PD 150606

£85.00 10mg

Calpain inhibitor.

PD 150606 is a cell-permeable non-peptide calpain inhibitor with Ki values for ν and m-calpains of 0.21 and 0.37 M. PD 150606 targets the calcium binding sites of calpain and possesses very high selectivity for calpains relative to other proteases, acting as a non-competitive inhibitor with regard to the substrate.

Please contact us for availability.

SKU: PI-110 Categories: ,

Additional information

Three Letter Sequence

Z-3-4-Iodophenyl-2-mercapto-2-propenoic acid

Molecular Weight

306.12

Molecular Formula

C9H7IO2S

Sequence

Z-3-4-Iodophenyl-2-mercapto-2-propenoic acid

Solubility

Soluble in DMSO and ethanol

Appearance

Off white solid

Storage

Store desiccated, frozen and in the dark

Purity

‰¥95% (HPLC)