BQ 3020

£125.00 1mg

SKU: ER-010 Categories: ,

Selective ETB receptor agonist.

BQ 3020 is a linear analogue of endothelin-1 (ET-1) which is a highly potent and selective ETB endothelin receptor agonist with Ki values of 0.18 and 970 nM at human ETB and ETA receptors. Intratumour administration of BQ 3020 can attenuate cancer pain by modulating ?-endorphin release from squamous cell carcinoma cells in mouse models.

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Additional information

Three Letter Sequence

Ac-Leu-Met-Asp-Lys-Glu-Ala-Val-Tyr-Phe-Ala-His-Leu-Asp-Ile-Ile-Trp-OH

Molecular Weight

2006.35

Molecular Formula

C96H140N20O25S

Sequence

Ac-LMDKEAVYFAHLDIIW

Solubility

Soluble to 0.50 mg/ml in sodium bicarbonate (0.03M)

Appearance

Freeze dried solid

Storage

Store dry, frozen and in the dark

Purity

>95% by HPLC

Modifications

N terminal acetyl

Searchable Words

BQ-3020, BQ3020, 143113-45-5, Ac-LMDKEAVYFAHLDIIW, LMDKEAVYFAHLDIIW